Publications
Found 23 results
Author [ Title] Type Year Filters: First Letter Of Last Name is E [Clear All Filters]
7-(2-Thienyl)-7-Deazaadenosine (AB61), a New Potent Nucleoside Cytostatic with a Complex Mode of Action. Molecular Cancer Therapeutics 2016, 15 (5), 922-937 DOI: 10.1158/1535-7163.MCT-14-0933.
Antiviral Activity of 7-Substituted 7-Deazapurine Ribonucleosides, Monophosphate Prodrugs, and Triphoshates against Emerging RNA Viruses. ACS Infectious Diseases 2021, 7 (2), 471-478.
Conversion of Thebaine to Oripavine and Other Useful Intermediates for the Semisynthesis of Opiate-Derived Agents: Synthesis of Hydromorphone. Advanced Synthesis & Catalysis 2014, 356 (11-12), 2679-2687 DOI: 10.1002/adsc.201400445.
Direct Synthesis of Noroxymorphone from Thebaine: Unusual Ce IV Oxidation of a Methoxydiene-Iron Complex to an Enone-γ-Nitrate. European Journal of Organic Chemistry 2016, 2016 (8), 1500-1503 DOI: 10.1002/ejoc.201600153.
Efficacy of the acyclic nucleoside phosphonates (S)-9-(3-fluoro-2-phosphonylmethoxypropyl)adenine (FPMPA) and 9-(2-phosphonylmethoxyethyl)adenine (PMEA) against feline immunodeficiency virus. Journal of Acquired Immune Deficiency Syndromes and Human Retrovirology 1998, 17 (2), 120-128.
Exploring the "Goldilocks Zone" of Semiconducting Polymer Photocatalysts by Donor-Acceptor Interactions. Angewandte Chemie-International Edition 2018, 57 (43), 14188-14192 DOI: 10.1002/anie.201809702.
Improved Synthesis of Buprenorphine from Thebaine and/or Oripavine via Palladium-Catalyzed N-Demethylation/Acylation and/or Concomitant O-Demethylation. Advanced Synthesis & Catalysis 2012, 354 (4), 613-626 DOI: 10.1002/adsc.201100807.
Labelling of nucleosides and oligonucleotides by solvatochromic 4-aminophthalimide fluorophore for studying DNA–protein interactions. Chemical Science 2012, 3 (9), 2797 DOI: 10.1039/c2sc20404e.
A Novel Bifunctional Allyldisilane as a Triple Allylation Reagent in the Stereoselective Synthesis of Trisubstituted Tetrahydrofurans. Chemistry - A European Journal 2011, 17 (26), 7162-7166 DOI: 10.1002/chem.201100513.
Oxidative DNA Cleavage with Clip-Phenanthroline Triplex-Forming Oligonucleotide Hybrids. Chembiochem : a European journal of chemical biology 2020, 21 (7), 991-1000 DOI: 10.1002/cbic.201900670.
Perfluoroalkylation through Cross-Metathesis between Alkenes and (Perfluoroalkyl)propenes. European Journal of Organic Chemistry 2008, 2008 (26), 4493-4499 DOI: 10.1002/ejoc.200800230.
Synthesis and Biochemical Characterization of a Series of 17α-Perfluoroalkylated Estradiols as Selective Ligands for Estrogen Receptor α. Journal of Medicinal Chemistry 2010, 53 (19), 6947-6953 DOI: 10.1021/jm100563h.
Synthesis and Cytostatic and Antiviral Activities of 2′-Deoxy-2′,2′-difluororibo- and 2′-Deoxy-2′-fluororibonucleosides Derived from 7-(Het)aryl-7-deazaadenines. ChemMedChem 2013, 8 (5), 832-846 DOI: 10.1002/cmdc.201300047.
Synthesis and evaluation of 17α-(carboranylalkyl)estradiols as ligands for estrogen receptors α and β. Journal of Organometallic Chemistry 2013, 747, 178-183 DOI: 10.1016/j.jorganchem.2013.06.013.
Synthesis of 2,6-disubstituted pyridin-3-yl C-2′-deoxyribonucleosides through chemoselective transformations of bromo-chloropyridine C-nucleosides. Organic & Biomolecular Chemistry 2013, 11 (28), 4702 DOI: 10.1039/c3ob40774h.
Synthesis of Fluorinated Brassinosteroids Based on Alkene Cross-Metathesis and Preliminary Biological Assessment. Journal of Medicinal Chemistry 2009, 52 (18), 5753-5757 DOI: 10.1021/jm900495f.
Synthesis of Mono(perfluoroalkyl) Cyclodextrins via Cross Metathesis. European Journal of Organic Chemistry 2010, 2010 (32), 6256-6262 DOI: 10.1002/ejoc.201000807.
Synthesis of Nororipavine and Noroxymorphone via N- and O-Demethylation of Iron Tricarbonyl Complex of Thebaine. Synthesis 2016, 48 (12), e1-e1 DOI: 10.1055/s-0035-1562345.
Synthesis of Perfluoroalkylated Carboranes by Cross-Metathesis of Allylcarboranes and Perfluoroalkylpropenes. Synlett 2010, 2010 (06), 885-888 DOI: 10.1055/s-0029-1219546.
Total synthesis of 4-F3t-neuroprostane and its 4-epimer. Tetrahedron Letters 2009, 50 (13), 1498-1500 DOI: 10.1016/j.tetlet.2009.01.075.
Transition-Metal-Mediated or -Catalyzed Syntheses of Steroids and Steroid-Like Compounds. European Journal of Organic Chemistry 2012, 2012 (1), 29-42 DOI: 10.1002/ejoc.201100921.
Twinned Growth of Metal-Free, Triazine-Based Photocatalyst Films as Mixed-Dimensional (2D/3D) van der Waals Heterostructures. Advanced Materials 2017, 29 (40), 1703399 DOI: 10.1002/adma.201703399.
Unexpected N -Demethylation of Oxymorphone and Oxycodone N -Oxides Mediated by the Burgess Reagent: Direct Synthesis of Naltrexone, Naloxone, and Other Antagonists from Oxymorphone. Advanced Synthesis & Catalysis 2012, 354 (14-15), 2706-2712 DOI: 10.1002/adsc.201200676.