Publications
Structure-based design and modular synthesis of novel PI4K class II inhibitors bearing a 4-aminoquinazoline scaffold. Bioorganic and Medicinal Chemistry Letters 2022, 76 (November), nestránkováno.
Structure-Aided Design of Novel Inhibitors of HIV Protease Based on a Benzodiazepine Scaffold. Journal of Medicinal Chemistry 2012, 55 (22), 10130-10135 DOI: 10.1021/jm301249q.
Structural characterization of the interaction between the C-terminal domain of the influenza polymerase PA subunit and an optimized small peptide inhibitor. Antiviral Research 2021, 185 (January), nestránkováno.
Structural Basis for Inhibition of Mycobacterial and Human Adenosine Kinase by 7-Substituted 7-(Het)aryl-7-deazaadenine Ribonucleosides. Journal of Medicinal Chemistry 2014, 57 (20), 8268-8279 DOI: 10.1021/jm500497v.
Sterically-Controlled Self-Immolation in Phosphoramidate Linkers Triggered by Light. European Journal of Organic Chemistry 2020, 2020 (7), 897-906 DOI: 10.1002/ejoc.201901882.
Stereoselective synthesis of (Z)-β-enamido fluorides from N-fluoroalkyl- and N-sulfonyl-1,2,3-triazoles. Organic Letters 2021, 23 (11), 4224-4227.
Stereoselective Synthesis of (Z)-beta-Enamido Triflates and Fluorosulfonates from N-Fluoroalkylated Triazoles. Chemistry-a European Journal 2019, 25 (32), 7640-7644 DOI: 10.1002/chem.201901632.
Stereoselective Synthesis of Ezetimibe via Cross-Metathesis of Homoallylalcohols and α-Methylidene-β-Lactams. The Journal of Organic Chemistry 2016, 81 (17), 7692-7699 DOI: 10.1021/acs.joc.6b01406.
Stereoselective cyclopropanation of boron dipyrromethene (BODIPY) derivatives by an organocascade reaction. Advanced Synthesis and Catalysis 2022, 364 (5), 930-937.
Squaramate-Modified Nucleotides and DNA for Specific Cross-Linking with Lysine-Containing Peptides and Proteins. Angewandte Chemie-International Edition 2019, 58 (38), 13345-13348 DOI: 10.1002/anie.201906737.
Spin-State-Controlled Photodissociation of Iron(III) Azide to an Iron(V) Nitride Complex. Angewandte Chemie-International Edition 2017, 56 (45), 14057-14060 DOI: 10.1002/anie.201707420.
Sphingosine and clavaminol H derivatives bearing fluorinated chains and their cytotoxic activity. Journal of Fluorine Chemistry 2012, 141, 49-57 DOI: 10.1016/j.jfluchem.2012.06.005.
Spectroscopic Characterization and Reactivity of Triplet and Quintet Iron(IV) Oxo Complexes in the Gas Phase. Angewandte Chemie International Edition 2016, 55 (11), 3637-3641 DOI: 10.1002/anie.201511374.
Specific Inhibitors of HIV Capsid Assembly Binding to the C-Terminal Domain of the Capsid Protein: Evaluation of 2-Arylquinazolines as Potential Antiviral Compounds. Journal of Medicinal Chemistry 2016, 59 (2), 545-558 DOI: 10.1021/acs.jmedchem.5b01089.
Speciation Behavior of Copper(II) Acetate in Simple Organic Solvents - Revealing the Effect of Trace Water: Speciation Behavior of Cu(II) Acetate in Simple Organic Solvents. European Journal of Inorganic Chemistry 2014, 2014 (8), 1407-1412 DOI: 10.1002/ejic.201400036.
Sonogashira reactions of α- and β-1-ethynyl-2-deoxyribosides: synthesis of acetylene-extended C-nucleosides. Tetrahedron 2010, 66 (2), 530-536 DOI: 10.1016/j.tet.2009.11.030.
Solvatochromic fluorene-linked nucleoside and DNA as color-changing fluorescent probes for sensing interactions. Chem. Sci. 2016, 7 (9), 5775-5785 DOI: 10.1039/C6SC02548J.
Solid-phase recombinase polymerase amplification using ferrocene-labelled dNTPs for electrochemical detection of single nucleotide polymorphisms. Biosensors and Bioelectronics 2022, 198 (February), nestránkováno.
Simple Preparation of 3(I)-O-Substituted β-Cyclodextrin Derivatives Using Cinnamyl Bromide. The Journal of Organic Chemistry 2005, 70 (22), 9054-9055 DOI: 10.1021/jo051339c.
A Simple Approach to Unsymmetric Atropoisomeric BipyridineN,N′-Dioxides and Their Application in Enantioselective Allylation of Aldehydes. Advanced Synthesis & Catalysis 2007, 349 (6), 822-826 DOI: 10.1002/adsc.200600400.
Simple and Fast Synthesis of New Axially Chiral Bipyridine N,N′ -Dioxides for Highly Enantioselective Allylation of Aldehydes. Advanced Synthesis & Catalysis 2009, 351 (9), 1279-1283 DOI: 10.1002/adsc.200900224.
Short Chemoenzymatic Azide-Free Synthesis of Oseltamivir (Tamiflu): Approaching the Potential for Process Efficiency. Advanced Synthesis & Catalysis 2010, 352 (1), 195-200 DOI: 10.1002/adsc.200900844.
Several Generations of Chemoenzymatic Synthesis of Oseltamivir (Tamiflu): Evolution of Strategy, Quest for a Process-Quality Synthesis, and Evaluation of Efficiency Metrics. The Journal of Organic Chemistry 2011, 76 (24), 10050-10067 DOI: 10.1021/jo2018872.
Separation of cyclodextrins and their derivatives by thin-layer and preparative column chromatography. Carbohydrate Research 1995, 275 (1), 1-7.
Sensitive CE-MS method for monitoring of riociguat and desmethylriociguat levels in human serum. Electrophoresis 2020, 41 (18-19), 1564-1567 DOI: 10.1002/elps.202000135.