Publications
Synthesis and evaluation of 17α-(carboranylalkyl)estradiols as ligands for estrogen receptors α and β. Journal of Organometallic Chemistry 2013, 747, 178-183 DOI: 10.1016/j.jorganchem.2013.06.013.
Synthesis, Molecular Structure, and Electrochemistry of 1-Ferrocenyl-1,2-dicarba- closo -dodecaboranes. European Journal of Inorganic Chemistry 2013, 2013 (15), 2789-2798 DOI: 10.1002/ejic.201300110.
Synthesis of 1,2,3,4-Tetramethyl- and 1,2,3,4-Tetraethylfluorene through a Dewar Benzene Pathway: Synthesis of 1,2,3,4-Tetramethyl- and 1,2,3,4-Tetraethylfluorene. European Journal of Organic Chemistry 2013, 2013 (1), 44-47 DOI: 10.1002/ejoc.201201343.
Synthesis of 2,6-disubstituted pyridin-3-yl C-2′-deoxyribonucleosides through chemoselective transformations of bromo-chloropyridine C-nucleosides. Organic & Biomolecular Chemistry 2013, 11 (28), 4702 DOI: 10.1039/c3ob40774h.
Synthesis of nucleosides and dNTPs bearing oligopyridine ligands linked through an octadiyne tether, their incorporation into DNA and complexation with transition metal cations. Org. Biomol. Chem. 2013, 11 (1), 78-89 DOI: 10.1039/C2OB26881G.
Sphingosine and clavaminol H derivatives bearing fluorinated chains and their cytotoxic activity. Journal of Fluorine Chemistry 2012, 141, 49-57 DOI: 10.1016/j.jfluchem.2012.06.005.
Structure-Aided Design of Novel Inhibitors of HIV Protease Based on a Benzodiazepine Scaffold. Journal of Medicinal Chemistry 2012, 55 (22), 10130-10135 DOI: 10.1021/jm301249q.
Sugar-modified derivatives of cytostatic 7-(het)aryl-7-deazaadenosines: 2′-C-methylribonucleosides, 2′-deoxy-2′-fluoroarabinonucleosides, arabinonucleosides and 2′-deoxyribonucleosides. Bioorganic & Medicinal Chemistry 2012, 20 (17), 5202-5214 DOI: 10.1016/j.bmc.2012.07.003.
Synthesis and antiviral activity of 4,6-disubstituted pyrimido[4,5-b]indole ribonucleosides. Bioorganic & Medicinal Chemistry 2012, 20 (20), 6123-6133 DOI: 10.1016/j.bmc.2012.08.021.
Synthesis of 2′-deoxy-2′-fluororibo- and 2′-deoxy-2′,2′-difluororibonucleosides derived from 6-(het)aryl-7-deazapurines. Tetrahedron 2012, 68 (39), 8300-8310 DOI: 10.1016/j.tet.2012.07.033.
Synthesis of 3I-O and 2I-O-monosubstituted derivatives of per-6-azido-β-cyclodextrin—potential molecular scaffolds. Carbohydrate Research 2012, 361, 148-154 DOI: 10.1016/j.carres.2012.09.003.
Synthesis of 6-Substituted 2(1H)-Pyridon-3-yl C-2′-Deoxyribonucleosides. European Journal of Organic Chemistry 2012, 2012 (9), 1759-1767 DOI: 10.1002/ejoc.201101662.
Synthesis of Aldehyde-Linked Nucleotides and DNA and Their Bioconjugations with Lysine and Peptides through Reductive Amination. Chemistry - A European Journal 2012, 18 (13), 4080-4087 DOI: 10.1002/chem.201103270.
Synthesis of Aromatic Compounds by Catalytic C-C Bond Activation of Biphenylene or Angular [3]Phenylene. Chemistry - A European Journal 2012, 18 (14), 4200-4207 DOI: 10.1002/chem.201103888.
Synthesis of Ferrocenestrone: the First Metallocene Based Steroid Analogue. Chemistry - A European Journal 2012, 18 (18), 5515-5518 DOI: 10.1002/chem.201200687.
Synthesis of Hydrazone-Modified Nucleotides and Their Polymerase Incorporation onto DNA for Redox Labeling. ChemPlusChem 2012, 77 (8), 652-662 DOI: 10.1002/cplu.201200056.
Synthesis of Substituted Benzyl Homo-C-Ribonucleosides and -Nucleotides as Carba Analogues of Phosphoribosylanthranilate. European Journal of Organic Chemistry 2012, 2012 (26), 4969-4981 DOI: 10.1002/ejoc.201200819.
Several Generations of Chemoenzymatic Synthesis of Oseltamivir (Tamiflu): Evolution of Strategy, Quest for a Process-Quality Synthesis, and Evaluation of Efficiency Metrics. The Journal of Organic Chemistry 2011, 76 (24), 10050-10067 DOI: 10.1021/jo2018872.
Supramolecular Engineering of Intrinsic and Extrinsic Porosity in Covalent Organic Cages. Journal of the American Chemical Society 2011, 133 (41), 16566-16571 DOI: 10.1021/ja2056374.
Synthesis and biological activity of desmethoxy analogues of coruscanone A. Bioorganic & Medicinal Chemistry Letters 2011, 21 (20), 6062-6066 DOI: 10.1016/j.bmcl.2011.08.059.
Synthesis of Buprenorphine from Oripavine via N-Demethylation of Oripavine Quaternary Salts. The Journal of Organic Chemistry 2011, 76 (11), 4628-4634 DOI: 10.1021/jo200567n.
Synthesis of Substituted Linear Ter- and Quaterphenyls via Dewar Benzenes. Synlett 2011, 2011 (03), 396-398 DOI: 10.1055/s-0030-1259321.
Short Chemoenzymatic Azide-Free Synthesis of Oseltamivir (Tamiflu): Approaching the Potential for Process Efficiency. Advanced Synthesis & Catalysis 2010, 352 (1), 195-200 DOI: 10.1002/adsc.200900844.
Sonogashira reactions of α- and β-1-ethynyl-2-deoxyribosides: synthesis of acetylene-extended C-nucleosides. Tetrahedron 2010, 66 (2), 530-536 DOI: 10.1016/j.tet.2009.11.030.
Synthesis and Biochemical Characterization of a Series of 17α-Perfluoroalkylated Estradiols as Selective Ligands for Estrogen Receptor α. Journal of Medicinal Chemistry 2010, 53 (19), 6947-6953 DOI: 10.1021/jm100563h.