Publications

Found 212 results
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2023
Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.
Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.
Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.
Holovko-Kamoshenkova, O. M.; Slivka, M. V.; Hrdina, R.; Baumer, V. N.; Korol, N. I.; Sokolenko, L. V.; Lendel, V. G. An Efficient Catalyst-Free Direct Approach to 5-Polyfluoroalkyl-1,2,4-triazole-3-thiones. Synthesis 2023, 55 (08), 1221-1226.
Belhajová, M.; Vícha, A.; Burgert, L.; Brožková, I.; Michaličková, L.; Hrdina, R.; Moravec, T.; Netuka, D.; Musil, Z.; Hrdina, R. En route to local glioblastoma treatment with temozolomide doped hyaluronan fibres: formulation and in vitro cell studies. RSC Medicinal Chemistry 2023, 14 (9), 1662-1666.
Belhajová, M.; Vícha, A.; Burgert, L.; Brožková, I.; Michaličková, L.; Hrdina, R.; Moravec, T.; Netuka, D.; Musil, Z.; Hrdina, R. En route to local glioblastoma treatment with temozolomide doped hyaluronan fibres: formulation and in vitro cell studies. RSC Medicinal Chemistry 2023, 14 (9), 1662-1666.
Belhajová, M.; Vícha, A.; Burgert, L.; Brožková, I.; Michaličková, L.; Hrdina, R.; Moravec, T.; Netuka, D.; Musil, Z.; Hrdina, R. En route to local glioblastoma treatment with temozolomide doped hyaluronan fibres: formulation and in vitro cell studies. RSC Medicinal Chemistry 2023, 14 (9), 1662-1666.
Nigríni, M.; Bhosale, V. Anandrao; Císařová, I.; Veselý, J. Enantioenriched 1,4-Benzoxazepines via Chiral Brønsted Acid-Catalyzed Enantioselective Desymmetrization of 3-Substituted Oxetanes. Journal of Organic Chemistry 2023, 88 (24), 17024-17036.
Misehe, M.; Matoušová, M.; Dvořáková, A.; Hercík, K.; Škach, K.; Chalupská, D.; Dejmek, M.; Šála, M.; Hájek, M.; Bouřa, E.; et al. Exploring positions 6 and 7 of a quinazoline-based scaffold leads to changes in selectivity and potency towards RIPK2/3 kinases. European Journal of Medicinal Chemistry 2023, 260 (November).
Ortiz, M.; Jauset-Rubio, M.; Trummer, O.; Foessl, I.; Kodr, D.; Acero, J. Lluís; Botero, M. Luz; Biggs, P.; Lenartowicz, D.; Trajanoska, K.; et al. Generic Platform for the Multiplexed Targeted Electrochemical Detection of Osteoporosis-Associated Single Nucleotide Polymorphisms Using Recombinase Polymerase Solid-Phase Primer Elongation and Ferrocene-Modified Nucleoside Triphosphates. ACS Central Science 2023, 9 (8), 1591-1602.
Ortiz, M.; Jauset-Rubio, M.; Trummer, O.; Foessl, I.; Kodr, D.; Acero, J. Lluís; Botero, M. Luz; Biggs, P.; Lenartowicz, D.; Trajanoska, K.; et al. Generic Platform for the Multiplexed Targeted Electrochemical Detection of Osteoporosis-Associated Single Nucleotide Polymorphisms Using Recombinase Polymerase Solid-Phase Primer Elongation and Ferrocene-Modified Nucleoside Triphosphates. ACS Central Science 2023, 9 (8), 1591-1602.
Janecký, L.; Markos, A.; Klepetářová, B.; Beier, P. Lewis-Acid-Mediated Intramolecular Cyclization of 4-Aryl-5-allyl-1,2,3-triazoles to Substituted Cyclopentene Derivatives. Journal of Organic Chemistry 2023, 88 (2), 1155-1167.
Navrátil, R.; Kellovská, K.; Baszczyňski, O. Multimetallic Pd- and Ni-catalyzed C(sp2)–P cross-coupling under aqueous micellar conditions. Green Chemistry 2023, 25 (23), 9779-9794.
Bakhanovich, O.; Klepetářová, B.; Beier, P. Rhodium(II)-catalyzed transannulation approach to N-fluoroalkylated indoles. Organic and Biomolecular Chemistry 2023, 21 (39), 7924-7927.
Bakhanovich, O.; Klepetářová, B.; Beier, P. Rhodium(II)-catalyzed transannulation approach to N-fluoroalkylated indoles. Organic and Biomolecular Chemistry 2023, 21 (39), 7924-7927.
Vrkoslav, V.; Horká, P.; Jindřich, J.; Buděšínský, M.; Cvačka, J. Silver Ion High-Performance Liquid Chromatography — Atmospheric Pressure Chemical Ionization Mass Spectrometry: A Tool for Analyzing Cuticular Hydrocarbons. Molecules 2023, 28 (9).
Lončarić, D.; Movahedifar, F.; Štoček, J. Radek; Dračínský, M.; Cvačka, J.; Guan, S.; Bythell, B. J.; Císařová, I.; Masson, E.; Kaleta, J. Solvent-controlled formation of alkali and alkali-earth-secured cucurbituril/guest trimers. Chemical Science 2023, 14 (35), 9258-9266.
Kuprikova, N.; Ondruš, M.; Bednárová, L.; Fernández, M. Riopedre; Slavětínská, L. Poštová; Sýkorová, V.; Hocek, M. Superanionic DNA: enzymatic synthesis of hypermodified DNA bearing four different anionic substituents at all four nucleobases. Nucleic Acids Research 2023, 51 (21), 11428-11438.
Ziabko, M.; Klepetářová, B.; Beier, P. Synthesis of Azidodifluoromethyl Phenyl Sulfone and Its Use as a Synthetic Equivalent of the Azidodifluoromethyl Anion. Journal of Organic Chemistry 2023, 88 (11), 6939-6946.
Antal, R.; Staś, M.; Perdomo, S. M.; Štemberová, M.; Brůža, Z.; Matouš, P.; Kratochvíl, J.; Růžička, A.; Rulíšek, L.; Kuneš, J.; et al. Synthesis of highly polarized [3]dendralenes and their Diels-Alder reactions. Organic Chemistry Frontiers 2023, 10 (22), 5568-5578.
Dejmek, M.; Brázdová, A.; Otava, T.; Polidarová, M. Pimková; Klíma, M.; Smola, M.; Vavřina, Z.; Buděšínský, M.; Dračínský, M.; Liboska, R.; et al. Vinylphosphonate-based cyclic dinucleotides enhance STING-mediated cancer immunotherapy. European Journal of Medicinal Chemistry 2023, 259 (November).
Dejmek, M.; Brázdová, A.; Otava, T.; Polidarová, M. Pimková; Klíma, M.; Smola, M.; Vavřina, Z.; Buděšínský, M.; Dračínský, M.; Liboska, R.; et al. Vinylphosphonate-based cyclic dinucleotides enhance STING-mediated cancer immunotherapy. European Journal of Medicinal Chemistry 2023, 259 (November).
Dejmek, M.; Brázdová, A.; Otava, T.; Polidarová, M. Pimková; Klíma, M.; Smola, M.; Vavřina, Z.; Buděšínský, M.; Dračínský, M.; Liboska, R.; et al. Vinylphosphonate-based cyclic dinucleotides enhance STING-mediated cancer immunotherapy. European Journal of Medicinal Chemistry 2023, 259 (November).
Dejmek, M.; Brázdová, A.; Otava, T.; Polidarová, M. Pimková; Klíma, M.; Smola, M.; Vavřina, Z.; Buděšínský, M.; Dračínský, M.; Liboska, R.; et al. Vinylphosphonate-based cyclic dinucleotides enhance STING-mediated cancer immunotherapy. European Journal of Medicinal Chemistry 2023, 259 (November).
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