Publications

Bhosale, V. Anandrao; Císařová, I.; Kamlar, M.; Veselý, J. Catalytic asymmetric addition to cyclic N-acyl-iminium: Access to sulfone-bearing contiguous quaternary stereocenters. Chemical Communications 2022, 58 (71), 9942-9945.

Baszczyňski, O.; Černý, J.; Čmoková, A.; Grobárová, V.; Kolařík, M.; Procházková, E.; Slapničková, M.; Štěpánek, O.; Zíková, A. Piperazine-Modified Ketoconazole Derivatives Show Increased Activity against Fungal and Trypanosomatid Pathogens. ChemMedChem 2022, 17 (21), nestránkováno.

Bouřa, E.; Dejmek, M.; Chalupská, D.; Klíma, M.; Matoušová, M.; Mertlíková-Kaiserová, H.; Misehe, M.; Nencka, R.; Šála, M. Structure-based design and modular synthesis of novel PI4K class II inhibitors bearing a 4-aminoquinazoline scaffold. Bioorganic and Medicinal Chemistry Letters 2022, 76 (November), nestránkováno.

Benýšek, J.; Krečmerová, M.; Matoušová, M.; Kaiserová, H. Mertlíkov; Otmar, M.; Pohl, R.; Pomeisl, K.; Pomeislová, A.; Slavětínská, L. Poštová; Rubešová, P. 1,2,4-Thiadiazole acyclic nucleoside phosphonates as inhibitors of cysteine dependent enzymes cathepsin K and GSK-3β. Bioorganic & Medicinal Chemistry 2021, 32 (February), nestránkováno.

Břehová, P.; Česnek, M.; Dračínský, M.; Chaloupecká, E.; Janeba, Z.; Mertlíková-Kaiserová, H.; Skácel, J.; Soto-Velasquez, M. P.; Tloušťová, E.; Watts, V. J. Acyclic nucleoside phosphonates with 2-aminothiazole base as inhibitors of bacterial and mammalian adenylate cyclases. European Journal of Medicinal Chemistry 2021, 222 (October 15 2021), nestránkováno.

Bouřa, E.; Čížek, K.; Eyer, L.; Hocek, M.; Hodek, J.; Konkoľová, E.; Kozák, J.; Milisavljević, N.; Nencka, R.; Pohl, R.; et al. Antiviral Activity of 7-Substituted 7-Deazapurine Ribonucleosides, Monophosphate Prodrugs, and Triphoshates against Emerging RNA Viruses. ACS Infectious Diseases 2021, 7 (2), 471-478.

Bricout, H.; Caronia, E.; Galia, A.; Tichá, I. Chena; Jindřich, J.; Léger, B.; Menuel, S.; Monflier, É.; Noël, S.; Ponchel, A.; et al. Asymmetric hydrogenation of ethyl pyruvate over aqueous dispersed Pt nanoparticles stabilized by a cinchonidine-functionalized β-cyclodextrin. Catalysis Communications 2021, 150 (February), nestránkováno.

Beytlerová, N.; Mateus, M. Alexandre; Kotora, M.; Rýček, L. Catalytic Cyclotrimerization Pathway for Synthesis of Selaginpulvilins C and D: Scope and Limitations. Organic Letters 2021, 23 (12), 4511-4515.

Bělinová, T.; Beneš, H.; Groborz, O.; Heizer, T.; Herynek, V.; Hrubý, M.; Loukotová, L.; Raabová, H.; Švec, P. Direct Comparison of Analogous Amphiphilic Gradient and Block Polyoxazolines. Macromolecules 2021, 54 (17), 8182-8194.

Bělinová, T.; Beneš, H.; Groborz, O.; Heizer, T.; Herynek, V.; Hrubý, M.; Loukotová, L.; Raabová, H.; Švec, P. Direct Comparison of Analogous Amphiphilic Gradient and Block Polyoxazolines. Macromolecules 2021, 54 (17), 8182-8194.

Baszczyňski, O.; Dračínský, M.; Dvořáková, A.; Hodek, J.; Chalupský, K.; Janeba, Z.; Kalčic, F.; Kaiserová, H. Mertlíkov; Strmeň, T.; Šebestík, J.; et al. Discovery of Modified Amidate (ProTide) Prodrugs of Tenofovir with Enhanced Antiviral Properties. Journal of Medicinal Chemistry 2021, 64 (22), 16425-16449.

Beier, P.; Chvojka, T.; Janecký, L.; Klepetářová, B.; Markos, A.; Martínek, T.; Martinez-Seara, H. Haloalkenyl Imidoyl Halides as Multifacial Substrates in the Stereoselective Synthesis of N-Alkenyl Compounds. Advanced Synthesis and Catalysis 2021, 363 (13), 3258-3266.

Bednářová, E.; Kotora, M.; Malatinec, Š.; Tanaka, H. Highly Enantioselective Ring-Opening of meso-Epoxides with O- and N-Nucleophiles Catalyzed by a Chiral Sc(III)/bipyridine Complex. European Journal of Organic Chemistry 2021, 2021 (8), 1249-1257.

Bourassi, M.; Gaálová, J.; Izák, P.; Jindřich, J.; Kasal, P.; Ladewig, B. P.; Michel, M. Nafion membranes modified by cationic cyclodextrin derivatives for enantioselective separation. Separation and Purification Technology 2021, 266 (July), nestránkováno.

Baszczyňski, O.; Císařová, I.; Flieger, M.; Kolařík, M.; Kucherak, O.; Procházková, E.; Stodůlková, E.; Tošner, Z. NMR Structure Elucidation of Naphthoquinones from Quambalaria cyanescens. Journal of Natural Products 2021, 84 (1), 46-55.

Baszczyňski, O.; Cigáň, M.; Filo, J.; Májek, M.; Procházková, E.; Straka, M.; Šimon, P. Phosphate linkers with traceable cyclic intermediates for self-immolation detection and monitoring. Chemical Communications 2021, 57 (2), 211-214.

Baszczyňski, O.; Gallardo, M. García; Procházková, E.; Šimon, P.; Tichotová, M. Phosphate-Based Self-Immolative Linkers for Tuneable Double Cargo Release. Chemistry - A European Journal 2021, 27 (50), 12763-12775.

Beier, P.; Janecký, L.; Klepetářová, B.; Markos, A.; Pohl, R. Stereoselective synthesis of (Z)-β-enamido fluorides from N-fluoroalkyl- and N-sulfonyl-1,2,3-triazoles. Organic Letters 2021, 23 (11), 4224-4227.

Bažíková, E.; Císařová, I.; Jagtap, P. Ramling; Matoušová, E.; Nechaev, A.; Neumannová, J. Synthesis of fused 1,2-naphthoquinones with cytotoxic activity using a one-pot three-step reaction. Organic and Biomolecular Chemistry 2021, 19 (15), 3434-3440.

Bakhanovich, O.; Beier, P.; Khutorianskyi, V.; Motornov, V. Synthesis of N-perfluoroalkyl-3,4-disubstituted pyrroles by rhodium-catalyzed transannulation of N-fluoroalkyl-1,2,3-triazoles with terminal alkynes. Beilstein Journal of Organic Chemistry 2021, 17 (February 18 2021), 504-510.

Bakhanovich, O.; Beier, P.; Khutorianskyi, V.; Motornov, V. Synthesis of N-perfluoroalkyl-3,4-disubstituted pyrroles by rhodium-catalyzed transannulation of N-fluoroalkyl-1,2,3-triazoles with terminal alkynes. Beilstein Journal of Organic Chemistry 2021, 17 (February 18 2021), 504-510.

Brábek, J.; Černochová, Z.; Groborz, O.; Hrubý, M.; Kolouchová, K.; Rösel, D.; Starčuk, Z.; Škarková, A.; Šlouf, M.; Švec, P. Thermo- and ROS-Responsive Self-Assembled Polymer Nanoparticle Tracers for F-19 MRI Theranostics. Biomacromolecules 2021, 22 (6), 2325-2337.

Brunderová, M.; Hocek, M.; Ivancova, I.; Krömer, M.; Slavětínská, L. Poštová. 2-Formyl-dATP as Substrate for Polymerase Synthesis of Reactive DNA Bearing an Aldehyde Group in the Minor Groove. ChemPlusChem 2020, 85 (6), 1164-1170 DOI: 10.1002/cplu.202000287.

Bednářová, E.; Kotora, M.; Malatinec, Š. Applications of Bolm's Ligand in Enantioselective Synthesis. Molecules 2020, 25 (4), nestránkováno DOI: 10.3390/molecules25050958.

Brynda, J.; Fanfrlík, J.; Hadzima, M.; Hánová, I.; Horn, M.; Houštecká, R.; Lepšík, M.; Majer, P.; Mareš, M.; Mertlíková-Kaiserová, H.; et al. Biomimetic Macrocyclic Inhibitors of Human Cathepsin D: Structure-Activity Relationship and Binding Mode Analysis. Journal of Medicinal Chemistry 2020, 63 (4), 1576-1596 DOI: 10.1021/acs.jmedchem.9b01351.