Publications

Bourassi, M.; Gaálová, J.; Izák, P.; Jindřich, J.; Kasal, P.; Ladewig, B. P.; Michel, M. Nafion membranes modified by cationic cyclodextrin derivatives for enantioselective separation. Separation and Purification Technology 2021, 266 (July), nestránkováno.

Baszczyňski, O.; Císařová, I.; Flieger, M.; Kolařík, M.; Kucherak, O.; Procházková, E.; Stodůlková, E.; Tošner, Z. NMR Structure Elucidation of Naphthoquinones from Quambalaria cyanescens. Journal of Natural Products 2021, 84 (1), 46-55.

Gallardo, P. Güixens; Hocek, M.; Kraus, T.; Kuba, M.; Matyašovský, J.; Palágyi, A.; Pohl, R.; Tack, L. Nucleotides bearing aminophenyl- or aminonaphthyl-3-methoxychromone solvatochromic fluorophores for the enzymatic construction of DNA probes for the detection of protein-DNA binding. Organic and Biomolecular Chemistry 2021, 19 (45), 9966-9974.

Baszczyňski, O.; Cigáň, M.; Filo, J.; Májek, M.; Procházková, E.; Straka, M.; Šimon, P. Phosphate linkers with traceable cyclic intermediates for self-immolation detection and monitoring. Chemical Communications 2021, 57 (2), 211-214.

Baszczyňski, O.; Gallardo, M. García; Procházková, E.; Šimon, P.; Tichotová, M. Phosphate-Based Self-Immolative Linkers for Tuneable Double Cargo Release. Chemistry - A European Journal 2021, 27 (50), 12763-12775.

Kočovský, P.; Kuneš, J.; Kysilka, O.; Májek, M.; Maříková, J.; Matouš, P.; Pour, M.; Růžička, A. Reaction Outcome Critically Dependent on the Method of Workup: An Example from the Synthesis of 1-Isoquinolones. Journal of Organic Chemistry 2021, 86 (12), 8078-8088.

Beier, P.; Janecký, L.; Klepetářová, B.; Markos, A.; Pohl, R. Stereoselective synthesis of (Z)-β-enamido fluorides from N-fluoroalkyl- and N-sulfonyl-1,2,3-triazoles. Organic Letters 2021, 23 (11), 4224-4227.

Hejdánek, J.; Hodek, J.; Konvalinka, J.; Kožíšek, M.; Machara, A.; Pachl, P.; Radilová, K.; Řezáčová, P.; Weber, J. Structural characterization of the interaction between the C-terminal domain of the influenza polymerase PA subunit and an optimized small peptide inhibitor. Antiviral Research 2021, 185 (January), nestránkováno.

Doleželová, E.; Downey, A. Michael; Hocek, M.; Nguyen, V. Hai; Pohl, R.; Rožánková, S.; Slapničková, M.; Tichý, M.; Tloušťová, E.; Zíková, A. Synthesis and anti-trypanosomal activity of 3'-fluororibonucleosides derived from 7-deazapurine nucleosides. Bioorganic and Medicinal Chemistry Letters 2021, 40 (May 15 2021), nestránkováno.

Doleželová, E.; Džubák, P.; Gurská, S.; Hajdúch, M.; Hocek, M.; Krajczyk, A.; Milisavljević, N.; Perlíková, P.; Slavětínská, L. Poštová; Slapničková, M.; et al. Synthesis and Antitrypanosomal Activity of 6-Substituted 7-Methyl-7-deazapurine Nucleosides. ACS Infectious Diseases 2021, 7 (4), 917-926.

Konvalinka, J.; Kožíšek, M.; Kráľ, M.; Machara, A.; Majer, P.; Radilová, K.; Reiberger, R. Synthesis and In Vitro Evaluation of C-7 and C-8 Luteolin Derivatives as Influenza Endonuclease Inhibitors, 2021.

Císařová, I.; Henriksson, E.; Kamlar, M.; Malo, M.; Sunden, H. Synthesis of cis-Oriented Vicinal Diphenylethylenes through a Lewis Acid-Promoted Annulation of Oxotriphenylhexanoates. Journal of Organic Chemistry 2021, 86 (13), 8660-8671.

Bažíková, E.; Císařová, I.; Jagtap, P. Ramling; Matoušová, E.; Nechaev, A.; Neumannová, J. Synthesis of fused 1,2-naphthoquinones with cytotoxic activity using a one-pot three-step reaction. Organic and Biomolecular Chemistry 2021, 19 (15), 3434-3440.

Bakhanovich, O.; Beier, P.; Khutorianskyi, V.; Motornov, V. Synthesis of N-perfluoroalkyl-3,4-disubstituted pyrroles by rhodium-catalyzed transannulation of N-fluoroalkyl-1,2,3-triazoles with terminal alkynes. Beilstein Journal of Organic Chemistry 2021, 17 (February 18 2021), 504-510.

Hurný, D.; Malečková, A.; Štuka, Č.; Tonar, Z.; Vejražka, M. Ten evidence-based recommendations for higher education. Mefanet+ 2021: Cooperation on the effective use of technology in medical and healthcare education reflecting on the challenges of today, 2021, 13-13.

Brábek, J.; Černochová, Z.; Groborz, O.; Hrubý, M.; Kolouchová, K.; Rösel, D.; Starčuk, Z.; Škarková, A.; Šlouf, M.; Švec, P. Thermo- and ROS-Responsive Self-Assembled Polymer Nanoparticle Tracers for F-19 MRI Theranostics. Biomacromolecules 2021, 22 (6), 2325-2337.

Catanzano, O.; Conte, C.; Fraix, A.; Kalydi, E.; Kasal, P.; Payamifar, S.; Quaglia, F.; Seggio, M.; Sortino, S. Visible light-activatable cyclodextrin-conjugates for the efficient delivery of nitric oxide with fluorescent reporter and their inclusion complexes with betaxolol. New Journal of Chemistry 2021, 45 (19), 8449-8455.

Brunderová, M.; Hocek, M.; Ivancova, I.; Krömer, M.; Slavětínská, L. Poštová. 2-Formyl-dATP as Substrate for Polymerase Synthesis of Reactive DNA Bearing an Aldehyde Group in the Minor Groove. ChemPlusChem 2020, 85 (6), 1164-1170 DOI: 10.1002/cplu.202000287.

Hocek, M.; Matyašovský, J. 2-Substituted 2 '-deoxyinosine 5 '-triphosphates as substrates for polymerase synthesis of minor-groove-modified DNA and effects on restriction endonuclease cleavage. Organic and Biomolecular Chemistry 2020, 18 (2), 255-262 DOI: 10.1039/c9ob02502b.

Drastík, M.; Holas, O.; Hroch, M.; Hutníková, M.; Kašpar, M.; Kudová, E.; Mičuda, S.; Pandey, A. V.; Pávek, P.; Smutný, T.; et al. 3 beta-Isoobeticholic acid efficiently activates the farnesoid X receptor (FXR) due to its epimerization to 3 alpha-epimer by hepatic metabolism. Journal of Steroid Biochemistry and Molecular Biology 2020, 202 (September), nestránkováno DOI: 10.1016/j.jsbmb.2020.105702.

Císařová, I.; Formánek, B.; Tauchman, J.; Vesely, J. Access to Spirocyclic Benzothiophenones with Multiple Stereocenters via an Organocatalytic Cascade Reaction. Journal of Organic Chemistry 2020, 85 (13), 8510-8521 DOI: 10.1021/acs.joc.0c00882.

Bednářová, E.; Kotora, M.; Malatinec, Š. Applications of Bolm's Ligand in Enantioselective Synthesis. Molecules 2020, 25 (4), nestránkováno DOI: 10.3390/molecules25050958.

Brynda, J.; Fanfrlík, J.; Hadzima, M.; Hánová, I.; Horn, M.; Houštecká, R.; Lepšík, M.; Majer, P.; Mareš, M.; Mertlíková-Kaiserová, H.; et al. Biomimetic Macrocyclic Inhibitors of Human Cathepsin D: Structure-Activity Relationship and Binding Mode Analysis. Journal of Medicinal Chemistry 2020, 63 (4), 1576-1596 DOI: 10.1021/acs.jmedchem.9b01351.

Báječný, M.; Beneš, J.; Czernek, J.; Dunlop, D.; Francová, P.; Groborz, O.; Heizer, T.; Hobza, P.; Hrubý, M.; Kolouchová, K.; et al. Chelating Polymers for Hereditary Hemochromatosis Treatment. Macromolecular Bioscience 2020, 20 (12), nestránkováno DOI: 10.1002/mabi.202000254.

Kasireddy, S. Reddy; Míšek, J.; Nosek, V.; Tarallo, V. Development of a simple high-throughput assay for directed evolution of enantioselective sulfoxide reductases. Chemical Communications 2020, 56 (40), 5386-5388 DOI: 10.1039/d0cc01660h.