Publications

Found 264 results
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2023
Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.
Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.
Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.
Novotná, K.; Tenora, L.; Prchalová, E.; Paule, J.; Alt, J.; Veeravalli, V.; Lam, J.; Wu, Y.; Šnajdr, I.; Gori, S.; et al. Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-l-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery. Journal of Medicinal Chemistry 2023, 66 (22), 15493-15510.
Novotná, K.; Tenora, L.; Prchalová, E.; Paule, J.; Alt, J.; Veeravalli, V.; Lam, J.; Wu, Y.; Šnajdr, I.; Gori, S.; et al. Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-l-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery. Journal of Medicinal Chemistry 2023, 66 (22), 15493-15510.
Holovko-Kamoshenkova, O. M.; Slivka, M. V.; Hrdina, R.; Baumer, V. N.; Korol, N. I.; Sokolenko, L. V.; Lendel, V. G. An Efficient Catalyst-Free Direct Approach to 5-Polyfluoroalkyl-1,2,4-triazole-3-thiones. Synthesis 2023, 55 (08), 1221-1226.
Holovko-Kamoshenkova, O. M.; Slivka, M. V.; Hrdina, R.; Baumer, V. N.; Korol, N. I.; Sokolenko, L. V.; Lendel, V. G. An Efficient Catalyst-Free Direct Approach to 5-Polyfluoroalkyl-1,2,4-triazole-3-thiones. Synthesis 2023, 55 (08), 1221-1226.
Spampinato, A.; Kužmová, E.; Pohl, R.; Sýkorová, V.; Vrábel, M.; Kraus, T.; Hocek, M. trans-Cyclooctene- and Bicyclononyne-Linked Nucleotides for Click Modification of DNA with Fluorogenic Tetrazines and Live Cell Metabolic Labeling and Imaging. Bioconjugate Chemistry 2023, 34 (4), 772-780.
Spampinato, A.; Kužmová, E.; Pohl, R.; Sýkorová, V.; Vrábel, M.; Kraus, T.; Hocek, M. trans-Cyclooctene- and Bicyclononyne-Linked Nucleotides for Click Modification of DNA with Fluorogenic Tetrazines and Live Cell Metabolic Labeling and Imaging. Bioconjugate Chemistry 2023, 34 (4), 772-780.
Misehe, M.; Matoušová, M.; Dvořáková, A.; Hercík, K.; Škach, K.; Chalupská, D.; Dejmek, M.; Šála, M.; Hájek, M.; Bouřa, E.; et al. Exploring positions 6 and 7 of a quinazoline-based scaffold leads to changes in selectivity and potency towards RIPK2/3 kinases. European Journal of Medicinal Chemistry 2023, 260 (November).
Misehe, M.; Matoušová, M.; Dvořáková, A.; Hercík, K.; Škach, K.; Chalupská, D.; Dejmek, M.; Šála, M.; Hájek, M.; Bouřa, E.; et al. Exploring positions 6 and 7 of a quinazoline-based scaffold leads to changes in selectivity and potency towards RIPK2/3 kinases. European Journal of Medicinal Chemistry 2023, 260 (November).
Osifová, Z.; Šála, M.; Dračínský, M. Hydrogen-Bonding Interactions of 8-Substituted Purine Derivatives. ACS Omega 2023, 8 (28), 25538-25548.
Kugler, M.; Hadzima, M.; Dzijak, R.; Rampmaier, R.; Srb, P.; Vrzal, L.; Voburka, Z.; Majer, P.; Řezáčová, P.; Vrábel, M. Identification of specific carbonic anhydrase inhibitors via in situ click chemistry, phage-display and synthetic peptide libraries: comparison of the methods and structural study. RSC Medicinal Chemistry 2023, 14 (1), 144-153.
Novotná, K.; Thomas, A. G.; Štěpánek, O.; Murphy, B.; Hin, N.; Skácel, J.; Mueller, L.; Tenora, L.; Pal, A.; Alt, J.; et al. Neutral sphingomyelinase 2 inhibitors based on the pyrazolo[1,5-a] scaffold. European Journal of Medicinal Chemistry 2023, 259 (November).
Novotná, K.; Thomas, A. G.; Štěpánek, O.; Murphy, B.; Hin, N.; Skácel, J.; Mueller, L.; Tenora, L.; Pal, A.; Alt, J.; et al. Neutral sphingomyelinase 2 inhibitors based on the pyrazolo[1,5-a] scaffold. European Journal of Medicinal Chemistry 2023, 259 (November).
Novotná, K.; Thomas, A. G.; Štěpánek, O.; Murphy, B.; Hin, N.; Skácel, J.; Mueller, L.; Tenora, L.; Pal, A.; Alt, J.; et al. Neutral sphingomyelinase 2 inhibitors based on the pyrazolo[1,5-a] scaffold. European Journal of Medicinal Chemistry 2023, 259 (November).
Socha, O.; Osifová, Z.; Dračínský, M. NMR-Challenge.com: An Interactive Website with Exercises in Solving Structures from NMR Spectra. Journal of Chemical Education 2023, 100 (2), 962-968.
Kodr, D.; Ortiz, M.; Sýkorová, V.; Yenice, C. Pinar; Lesnikowski, Z. J.; O’Sullivan, C. K.; Hocek, M. Normalized Multipotential Redox Coding of DNA Bases for Determination of Total Nucleotide Composition. Analytical Chemistry 2023, 95 (34), 12586-12589.
Runemark, A.; Martos, M.; Nigríni, M.; Noa, F. M. Amombo; Öhrström, L.; Sunden, H. Photochemical Access to Substituted β-Lactams and β-Lactones via the Zimmerman–O’Connell–Griffin Rearrangement. Organic Letters 2023, 25 (29), 5520-5524.
Štefek, M.; Chalupská, D.; Chalupský, K.; Zgarbová, M.; Dvořáková, A.; Krafčíková, P.; Li, A. Shi Ming; Šála, M.; Dejmek, M.; Otava, T.; et al. Rational Design of Highly Potent SARS-CoV-2 nsp14 Methyltransferase Inhibitors. ACS Omega 2023, 8 (30), 27410-27418.
Štefek, M.; Chalupská, D.; Chalupský, K.; Zgarbová, M.; Dvořáková, A.; Krafčíková, P.; Li, A. Shi Ming; Šála, M.; Dejmek, M.; Otava, T.; et al. Rational Design of Highly Potent SARS-CoV-2 nsp14 Methyltransferase Inhibitors. ACS Omega 2023, 8 (30), 27410-27418.
Mulholland, C.; Jestřábová, I.; Sett, A.; Ondruš, M.; Sýkorová, V.; C. Manzanares, L.; Šimončík, O.; Muller, P.; Hocek, M. The selection of a hydrophobic 7-phenylbutyl-7-deazaadenine-modified DNA aptamer with high binding affinity for the Heat Shock Protein 70. Communications Chemistry 2023, 6 (1).
Mulholland, C.; Jestřábová, I.; Sett, A.; Ondruš, M.; Sýkorová, V.; C. Manzanares, L.; Šimončík, O.; Muller, P.; Hocek, M. The selection of a hydrophobic 7-phenylbutyl-7-deazaadenine-modified DNA aptamer with high binding affinity for the Heat Shock Protein 70. Communications Chemistry 2023, 6 (1).
Mulholland, C.; Jestřábová, I.; Sett, A.; Ondruš, M.; Sýkorová, V.; C. Manzanares, L.; Šimončík, O.; Muller, P.; Hocek, M. The selection of a hydrophobic 7-phenylbutyl-7-deazaadenine-modified DNA aptamer with high binding affinity for the Heat Shock Protein 70. Communications Chemistry 2023, 6 (1).
Lončarić, D.; Movahedifar, F.; Štoček, J. Radek; Dračínský, M.; Cvačka, J.; Guan, S.; Bythell, B. J.; Císařová, I.; Masson, E.; Kaleta, J. Solvent-controlled formation of alkali and alkali-earth-secured cucurbituril/guest trimers. Chemical Science 2023, 14 (35), 9258-9266.
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