Publications

Found 184 results
Author Title Type [ Year(Desc)]
Filters: First Letter Of Last Name is P  [Clear All Filters]
2021
Hejdánek, J.; Hodek, J.; Konvalinka, J.; Kožíšek, M.; Machara, A.; Pachl, P.; Radilová, K.; Řezáčová, P.; Weber, J. Structural characterization of the interaction between the C-terminal domain of the influenza polymerase PA subunit and an optimized small peptide inhibitor. Antiviral Research 2021, 185 (January), nestránkováno.
Doleželová, E.; Downey, A. Michael; Hocek, M.; Nguyen, V. Hai; Pohl, R.; Rožánková, S.; Slapničková, M.; Tichý, M.; Tloušťová, E.; Zíková, A. Synthesis and anti-trypanosomal activity of 3'-fluororibonucleosides derived from 7-deazapurine nucleosides. Bioorganic and Medicinal Chemistry Letters 2021, 40 (May 15 2021), nestránkováno.
Doleželová, E.; Džubák, P.; Gurská, S.; Hajdúch, M.; Hocek, M.; Krajczyk, A.; Milisavljević, N.; Perlíková, P.; Slavětínská, L. Poštová; Slapničková, M.; et al. Synthesis and Antitrypanosomal Activity of 6-Substituted 7-Methyl-7-deazapurine Nucleosides. ACS Infectious Diseases 2021, 7 (4), 917-926.
Catanzano, O.; Conte, C.; Fraix, A.; Kalydi, E.; Kasal, P.; Payamifar, S.; Quaglia, F.; Seggio, M.; Sortino, S. Visible light-activatable cyclodextrin-conjugates for the efficient delivery of nitric oxide with fluorescent reporter and their inclusion complexes with betaxolol. New Journal of Chemistry 2021, 45 (19), 8449-8455.
2022
Dian, J.; Fourmentin, S.; Jindřich, J.; Palágyi, A. Cyclodextrin-based Schiff base pro-fragrances: Synthesis and release studies. Beilstein Journal of Organic Chemistry 2022, 18 (September), 1346-1354.
Císařová, I.; David, T.; Dračínský, M.; Jirák, D.; Jurok, R.; Kretschmer, J.; Kuchař, M.; Polášek, M.; Socha, O.; Vít, M. Paramagnetic encoding of molecules. Nature Communications [online] 2022, 13 (1), nestránkováno.
Baszczyňski, O.; Černý, J.; Čmoková, A.; Grobárová, V.; Kolařík, M.; Procházková, E.; Slapničková, M.; Štěpánek, O.; Zíková, A. Piperazine-Modified Ketoconazole Derivatives Show Increased Activity against Fungal and Trypanosomatid Pathogens. ChemMedChem 2022, 17 (21), nestránkováno.
2023
Vopálenská, A.; Dočekal, V.; Petrželová, S.; Císařová, I.; Veselý, J. Access to Spirooxindole-Fused Cyclopentanes via a Stereoselective Organocascade Reaction Using Bifunctional Catalysis. Journal of Organic Chemistry 2023, 88 (12), 7724-7735.
Ulč, J.; Jacko, J.; Císařová, I.; Pospíšil, L.; Nečas, D.; Kotora, M. Catalytic C−C/C−H Bond Activation Relay for Synthesis of Fluorescent Naphthoquinolizinium Salts. European Journal of Organic Chemistry 2023, 26 (18).
Prener, L.; Baszczyňski, O.; Kaiser, M. Maxmilian; Dračínský, M.; Stepan, G.; Lee, Y. - J.; Brumshtein, B.; Yu, H.; Jansa, P.; Lansdon, E. B.; et al. Design and Synthesis of Novel HIV-1 NNRTIs with Bicyclic Cores and with Improved Physicochemical Properties. Journal of Medicinal Chemistry 2023, 66 (3), 1761-1777.
Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.
Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.
Novotná, K.; Tenora, L.; Prchalová, E.; Paule, J.; Alt, J.; Veeravalli, V.; Lam, J.; Wu, Y.; Šnajdr, I.; Gori, S.; et al. Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-l-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery. Journal of Medicinal Chemistry 2023, 66 (22), 15493-15510.
Novotná, K.; Tenora, L.; Prchalová, E.; Paule, J.; Alt, J.; Veeravalli, V.; Lam, J.; Wu, Y.; Šnajdr, I.; Gori, S.; et al. Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-l-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery. Journal of Medicinal Chemistry 2023, 66 (22), 15493-15510.
Spampinato, A.; Kužmová, E.; Pohl, R.; Sýkorová, V.; Vrábel, M.; Kraus, T.; Hocek, M. trans-Cyclooctene- and Bicyclononyne-Linked Nucleotides for Click Modification of DNA with Fluorogenic Tetrazines and Live Cell Metabolic Labeling and Imaging. Bioconjugate Chemistry 2023, 34 (4), 772-780.
Kodr, D.; Kužmová, E.; Pohl, R.; Kraus, T.; Hocek, M. Lipid-linked nucleoside triphosphates for enzymatic synthesis of hydrophobic oligonucleotides with enhanced membrane anchoring efficiency. Chemical Science 2023, 14 (15), 4059-4069.
Novotná, K.; Thomas, A. G.; Štěpánek, O.; Murphy, B.; Hin, N.; Skácel, J.; Mueller, L.; Tenora, L.; Pal, A.; Alt, J.; et al. Neutral sphingomyelinase 2 inhibitors based on the pyrazolo[1,5-a] scaffold. European Journal of Medicinal Chemistry 2023, 259 (November).
Novotná, K.; Thomas, A. G.; Štěpánek, O.; Murphy, B.; Hin, N.; Skácel, J.; Mueller, L.; Tenora, L.; Pal, A.; Alt, J.; et al. Neutral sphingomyelinase 2 inhibitors based on the pyrazolo[1,5-a] scaffold. European Journal of Medicinal Chemistry 2023, 259 (November).
Kuba, M.; Pohl, R.; Kraus, T.; Hocek, M. Nucleotides Bearing Red Viscosity-Sensitive Dimethoxy-Bodipy Fluorophore for Enzymatic Incorporation and DNA Labeling. Bioconjugate Chemistry 2023, 34 (1), 133-139.
Antal, R.; Staś, M.; Perdomo, S. M.; Štemberová, M.; Brůža, Z.; Matouš, P.; Kratochvíl, J.; Růžička, A.; Rulíšek, L.; Kuneš, J.; et al. Synthesis of highly polarized [3]dendralenes and their Diels-Alder reactions. Organic Chemistry Frontiers 2023, 10 (22), 5568-5578.
Antal, R.; Staś, M.; Perdomo, S. M.; Štemberová, M.; Brůža, Z.; Matouš, P.; Kratochvíl, J.; Růžička, A.; Rulíšek, L.; Kuneš, J.; et al. Synthesis of highly polarized [3]dendralenes and their Diels-Alder reactions. Organic Chemistry Frontiers 2023, 10 (22), 5568-5578.
Lapinskaite, R.; Atalay, H. Nazlican; Malatinec, Š.; Dönmez, S.; Cinar, Z. Özlem; Schwarz, P. F.; Perhal, A. F.; Císařová, I.; Labanauskas, L.; Karpiński, T. M.; et al. Synthesis of Selagibenzophenone A and Its Derivatives for Evaluation of Their Antiproliferative, ROR gamma Inverse Agonistic, and Antimicrobial Effect. ChemistrySelect 2023, 8 (7).
Dejmek, M.; Brázdová, A.; Otava, T.; Polidarová, M. Pimková; Klíma, M.; Smola, M.; Vavřina, Z.; Buděšínský, M.; Dračínský, M.; Liboska, R.; et al. Vinylphosphonate-based cyclic dinucleotides enhance STING-mediated cancer immunotherapy. European Journal of Medicinal Chemistry 2023, 259 (November).
Díaz-Holguín, A.; Rashidian, A.; Pijnenburg, D.; Ferreira, G. Monteiro; Štefela, A.; Kašpar, M.; Kudová, E.; Poso, A.; van Beuningen, R.; Pávek, P.; et al. When Two Become One: Conformational Changes in FXR/RXR Heterodimers Bound to Steroidal Antagonists. ChemMedChem 2023, 18 (4).
Díaz-Holguín, A.; Rashidian, A.; Pijnenburg, D.; Ferreira, G. Monteiro; Štefela, A.; Kašpar, M.; Kudová, E.; Poso, A.; van Beuningen, R.; Pávek, P.; et al. When Two Become One: Conformational Changes in FXR/RXR Heterodimers Bound to Steroidal Antagonists. ChemMedChem 2023, 18 (4).
xs sm md lg