Publications

Machara, A.; Endoma-Arias, M. Ann A.; Císařová, I.; D. Cox, P.; Hudlicky, T. Direct Synthesis of Noroxymorph­one from Thebaine: Unusual Ce ^IV Oxidation of a Methoxydiene-Iron Complex to an Enone-γ-Nitrate. European Journal of Organic Chemistry 2016, 2016 (8), 1500-1503 DOI: 10.1002/ejoc.201600153.

Machara, A.; Endoma-Arias, M.; Císařová, I.; Cox, D.; Hudlicky, T. Synthesis of Nororipavine and Noroxymorphone via N- and O-Demethylation of Iron Tricarbonyl Complex of Thebaine. Synthesis 2016, 48 (12), e1-e1 DOI: 10.1055/s-0035-1562345.

Machara, A.; Konvalinka, J.; Kotora, M. A MODULAR SYNTHESIS OF N -BENZOTRIAZOLE UREAS USING ALKYLATION OF 5-NITROBENZOTRIAZOLE. ChemistrySelect 2016, 1 (1), 101-107 DOI: 10.1002/slct.201600025.

Machara, A.; Lux, V.; Kožíšek, M.; Šašková, K. Grantz; Štěpánek, O.; Kotora, M.; Parkan, K.; Pávová, M.; Glass, B.; Sehr, P.; et al. Specific Inhibitors of HIV Capsid Assembly Binding to the C-Terminal Domain of the Capsid Protein: Evaluation of 2-Arylquinazolines as Potential Antiviral Compounds. Journal of Medicinal Chemistry 2016, 59 (2), 545-558 DOI: 10.1021/acs.jmedchem.5b01089.

Machara, A.; D. Cox, P.; Hudlicky, T. Direct Synthesis of Naltrexone by Palladium-Catalyzed N -Demethylation/Acylation of Oxymorphone: The Benefit of CH Activation and the Intramolecular Acyl Transfer from C-14 Hydroxy. Advanced Synthesis & Catalysis 2012, 354 (14-15), 2713-2718 DOI: 10.1002/adsc.201200677.

Machara, A.; Svoboda, J. Thiophenium-ylides: Synthesis and reactivity. Chemical Papers 2013, 67 (1) DOI: 10.2478/s11696-012-0222-7.

Machara, A.; Werner, L.; Endoma-Arias, M. Ann; D. Cox, P.; Hudlicky, T. Improved Synthesis of Buprenorphine from Thebaine and/or Oripavine via Palladium-Catalyzed N-Demethylation/Acylation and/or Concomitant O-Demethylation. Advanced Synthesis & Catalysis 2012, 354 (4), 613-626 DOI: 10.1002/adsc.201100807.

Machara, A.; D. Cox, P.; Hudlicky, T. ChemInform Abstract: Synthesis of Nalbuphine from Oripavine via N-Demethylation of N-Cyclobutylmethyl Oripavine. ChemInform 2012, 43 (19), no-no DOI: 10.1002/chin.201219209.

Machara, A.; Kozmík, V.; Pojarová, M.; Dvořáková, H.; Svoboda, J. Preparation and rearrangement study of novel thiophenium- and selenophenium-ylides. Collection of Czechoslovak Chemical Communications 2009, 1 DOI: 10.1135/cccc2009001.

Machara, A.; Pojarová, M.; Svoboda, J. Synthesis and Cycloaddition Reaction of 3-Vinylthieno[3,2-b][1]benzothiophene. Collection of Czechoslovak Chemical Communications 2007, 72 (7), 952-964 DOI: 10.1135/cccc20070952.

Machara, A.; Kurfürst, M.; Kozmı́k, V.; Petřı́čková, H.; Dvořáková, H.; Svoboda, J. A nonconcerted cycloaddition of fused 2-vinylthiophenes with dimethyl acetylenedicarboxylate. Tetrahedron Letters 2004, 45 (10), 2189-2192 DOI: 10.1016/j.tetlet.2004.01.030.